Synthesis of 4-hydroxyquinoline-2,3-dicarboxylates using N-(2-aminobenzoyl)benzotriazoles

ÇELİK İ., Yildiz F.

TETRAHEDRON, cilt.73, sa.27-28, ss.3878-3882, 2017 (SCI-Expanded) identifier identifier

  • Yayın Türü: Makale / Tam Makale
  • Cilt numarası: 73 Sayı: 27-28
  • Basım Tarihi: 2017
  • Doi Numarası: 10.1016/j.tet.2017.05.058
  • Dergi Adı: TETRAHEDRON
  • Derginin Tarandığı İndeksler: Science Citation Index Expanded (SCI-EXPANDED), Scopus, Index Chemicus (IC), Current Chemical Reactions (CCR)
  • Sayfa Sayıları: ss.3878-3882
  • Anahtar Kelimeler: Benzotriazole, 4-Hydroxyquinoline-2,3-dicarboxylate, N-(2-aminobenzoyl)benzotriazole, Annulation, Aza-Michael addition, INHIBITORS, MODEL
  • Anadolu Üniversitesi Adresli: Evet

Özet

A method for the preparation of 4-hydroxyquinoline-2,3-dicarboxylates has been developed by aza-Michael addition reaction of N-(2-aminobenzoyl)benzotriazoles with dimethyl acetylenedicarboxylate. 4-Hydroxyquinoline-2,3-dicarboxylates were obtained in moderate to good yields (53-87%). (C) 2017 Elsevier Ltd. All rights reserved.