A new protocol for the synthesis of primary, secondary and tertiary anthranilamides utilizing N-(2-aminoarylacyl)benzotriazoles

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KANIŞKAN N., Kokten S., ÇELİK İ.

ARKIVOC, cilt.2012, ss.198-213, 2012 (SCI-Expanded) identifier identifier

  • Yayın Türü: Makale / Tam Makale
  • Cilt numarası: 2012
  • Basım Tarihi: 2012
  • Doi Numarası: 10.3998/ark.5550190.0013.818
  • Dergi Adı: ARKIVOC
  • Derginin Tarandığı İndeksler: Science Citation Index Expanded (SCI-EXPANDED), Scopus
  • Sayfa Sayıları: ss.198-213
  • Anahtar Kelimeler: Anthranilic acid, benzotriazole, N-(2-aminoarylacyl)benzotrazoles, anthranilamides, BIOLOGICAL EVALUATION, N-ACYLBENZOTRIAZOLES, DERIVATIVES, INHIBITORS, RECEPTOR, IDENTIFICATION, BENZAMIDINES, CONVENIENT, EFFICIENT, ESTERS
  • Anadolu Üniversitesi Adresli: Evet

Özet

A convenient route for efficient conversion of unprotected anthranilic acids into the corresponding N-(2-aminoarylacyl)benzotrazoles is described. N-(2-Aminoarylacyl)benzotrazoles have been successfully used to synthesize primary, secondary and tertiary anthranilamides in high yields (71-96%).